Bredereck's reagent
BUJNO Synthesis Sp. z o. o.
Dorodna 16
03-195 Warszawa, POLAND

CAS: 5815-08-7 formula
FW: 174,28
Boiling point: 48-52oC, 10-12mm Hg

B1004 Bredereck reagent 98%
derivatisation grade
5 ml Price request
B985 Bredereck reagent 95%
50 ml Price request
B585 Bredereck reagent 90%
for synthesis
1000 ml
and 2500 ml
Price request
Purity confirmed by GC and NMR

  • Aminalester. Zur Stabilität und Umsetzung mit aromatischen Aldehydem
    Bredereck, H.; Simchen, G.; Hoffmann, H.; Horn, P.; Wahl, R.; Angew. Chem., 79 (1967) 311.
  • Darstellung und Eigenschaften der Amidacetale und Aminalester,
    Hellmut Bredereck, Gerhard Simchen, Siegfried Rebsdat, Willi Kantlehner, Peter Horn, Rudolf Wahl, Horst Hoffmann und Peter Grieshaber, Chem. Ber., 101 (1968) 41.
  • New synthetic reactions. Generalalkylation via a-trimetylenedithiocyclobutanones
    Trost, B.M.; Preckel, M.; J. Am. Chem. Soc.; 97 (1975) 2224.
  • A novel metod for converting ketones to a-diketones. The reaction of enamino ketones with singlet oxygen
    Wassermann, H.H.; Ives, J.L.; J. Am. Chem. Soc.; 98 (1976) 7868.
  • Asymmetric synthesis of allo-heteroyohimbine alkaloids
    Uskokovic, M.R.; Lewis, R.L.; Partridge, J.J.; Despreaux, C.W.; Pruess, D.L.; J. Am. Chem. Soc.; 101 (1979) 6742.
  • Orthoamide, XXXII. Umsetzungen von tert-Butoxy-N,N,N',N'-tetramethylmethandiamin mit NH- und CH-aciden Verbindungen
    Kantlehner, W.; Wagner, F.; Bredereck, H.; Liebigs Ann. Chem., (1980) 344.
  • Tetracarbonylferrate aus Orthoameisensäurederivaten und Pentacarbonyleisen
    Daub, J.; Hasenhündl, A.; Krenkler, K.P.; Schmetzer, J.; Liebigs Ann. Chem., (1980) 997.
  • Darstellung und Reaktionen von Trimethoxyacetamid und Trimethoxyacetamidderivaten
    Kantlehner, W.; Kapassakalidis, J.J.; Maier, T.; Liebigs Ann. Chem., (1980) 1448.
  • Synthesis of 2'-methylated pyrimidine C-nucleosides
    Sato, T.; Kobayashi, H.; Noyori, R.; Tetrahedron Lett., 21 (1980) 1971.
  • Synthesis of 4'-hydroxymethylated pyrimidine ribo-C-nucleosides
    Sato, T.; Noyori, R.; Tetrahedron Lett., 21 (1980) 2535.
  • Total synthesis of racemic ajmalicine and 19-epi-ajmalicine
    Gutzwiller, J.; Pizzolato, G.; Uskokovic, M.R.; Helv. Chim. Acta, 64 (1981) 1663.
  • Orthoamide, XXXVI. Zur Formylierung von 2,5-Dialkyl-1,3,4-thiadiazolen und 2,3,5-Trialkyl-1,3,4-thiadiazoliumsalzen durch Orthoamide der Ameisensäure
    Kantlehner, W.; Haug, E.; Hagen, H.; Liebigs Ann. Chem., (1982) 298.
  • Einfache Synthese von a-substituierten Tetronsäure-Derivaten
    Schmidt, R.R.; Betz, R.; Synthesis, (1982) 748.
  • Stereocontrolled general synthesis of pyrimidine C-nucleosides having branched-chain sugar moieties
    Sato, T.; Watanabe, M.; Kobayashi, H.; Noyori, R.; Bull. Chem. Soc. Jpn., 56 (1983) 2680.
  • Fungal metabolites. Part 15. Structure and chemical correlations of uvidin C, D, and E, new drimane sesquiterpenes from Lactarius uvidus Fries
    De Bernardi, M.; Mellerio, G.; Vidari, G.; Vita-Finzi, P.; Fronza, G.; J. Chem. Soc., Perkin Trans. 1, (1983) 2739.
  • Stereoselective synthesis of racemic trichodiene
    Schlessinger, R.H.; Schulz, J.A.; J. Org. Chem., 48 (1983) 407.
  • Synthetic strategies toward the synthesis of 2,4-dimethoxypyrrolo[3,2-d]pyrimidine
    Cupps, T.L.; Wise, D.S.; Townsend, L.B.; J. Org. Chem., 48 (1983) 1060.
  • Bromination of some pyridine and diazine N-oxides
    Paudler, W.W.; Jovanovic, M.V.; J. Org. Chem., 48 (1983) 1064.
  • Synthesis of porphyrinoctakis(dialkylcarboxamides)
    Kaesler, R.W.; LeGoff, E.; J. Org. Chem., 48 (1983) 4399.
  • Benz[c,d]indoles - I. The use of tert-buthoxy-bis-(dimethylamino)-methane
    Haeflinger, W.; Knecht, H.; Tetrahedron Lett., 24 (1983) 285.
  • Synthese de cyclopena[c]tetrahydropyridines precuseurs d'alcaloides monoterpeniques
    Brayer, J.-L.; Alazard, J.-P.; Thal, C.; Tetrahedron Lett., 24 (1983) 4193.
  • Reaction of singlet oxygen with enamino carbonyl systems. A general method for the synthesis of a-keto derivatives of lactones, esters, amides, lactams and ketonem
    Wassermann, H.H.; Ives, J.L.; J. Org. Chem., 50 (1985) 3573.
  • Simple enols. 4. Generation of some new simple enols in solution and the kinetics and mechanism of their ketonization
    Capon, B.; Siddhanta, A.K.; Zucco, C.; J. Org. Chem., 50 (1985) 3580.
  • O-Glycosylimidate, 19. Reaktionen von Glycosyl-trichloracetimidaten mit silylierten C-Nucleophilen
    Hoffmann, M.G.; Schmidt R.R.; Liebigs Ann. Chem., (1985) 2403.
  • Total synthesis of acosamine and daunosamine utilizing a diastereoselective intramolecular [3+2] cycloaddition
    Wovkulich, P.M.; Uskokovic, M.R.; Tetrahedron, 41 (1985) 3455.
  • An enantiospecific synthesis of estrone
    Hutchinson, J.H.; Money, T.; Tetrahedron Lett., 26 (1985) 1819.
  • New piperidinic synthons via ring contraction. Formal synthesis of (+/-)-perhydrohistrionicotoxin
    Duhamel, P.; Kotera, M.; Monteil, T.; Bull. Chem. Soc. Jpn., 56 (1986) 2353.
  • Reaktionen mit 2-aza-1,3-butadien-Derivaten, 1. Eine neue und besonders einfache Synthese von zentralaktiven b-Carbolin-Derivaten
    Biere, H.; Russe, R.; Seelen, W.; Liebigs Ann. Chem., (1986) 1749.
  • The synthesis of Mannich bases from ketonem and esters via enaminones
    Schuda, P.F.; Ebner, C.B.; Morgan, T.M.; Tetrahedron Lett., 27 (1986) 2567.
  • Enantiospecific synthesis of estrone
    Hutchinson, J.H.; Money, T.; Can. J. Chem., 65 (1987) 1.
  • Electron-rich and electron-poor pentalene derivatives
    Frank, W.; Gompper, R.; Tetrahedron Lett., 28 (1987) 3083.
  • Thermolysis of polyazapentadienes. Part 11. Concerted and free radical mechanisms in 2-aza enone and 2-aza enthione pyrolyses: crystal and molecular structures of 3-dimethylamino-1-p-tolyl-2-azaprop-2-en-1-one and 3-dimethylamino-1-phenyl-2-azaprop-2-ene-1-thione
    Blake, A.J.; McNab, H.; Murray, M.E.-A.; J. Chem. Soc., Perkin Trans. 1, (1989) 589.
  • New 7-substituted quinolone antibacterial agents. II. The synthesis of 1-ethyl-1,4-dihydro-4-oxo-7-(pyrazoyl, isoxazoyl, and pyrimidinyl)-1,8-naphthyridine and quinolone-3-carboxylic acids
    Domagala, J.M.; Peterson, P.; J. Heterocyclic Chem., 26 (1989) 1147.
  • Highly stereoselective ring contraction of heterocyclic enamines: total synthesis of perhydrohistrionicotoxin and its 2,6-epimer
    Duhamel, P.; Kotera, M.; Monteil, T.; Marabout, B.; J. Org. Chem., 54 (1989) 4419.
  • Total synthesis of ( )-jolkinolide A, B, and E utilizing a new mild estrification followed by intramolecular Wittig-Horner reaction
    Katsumura, S.; Kimura, A.; Isoe, S.; Tetrahedron, 45 (1989) 1337.
  • Tricyclic Pyridine Derivatives with High Affinity to the Central Benzodiazepine Receptor
    Fischer, U.; Möhler, H.; Schneider, F.; Widmer, U.; Helv. Chim. Acta, 73 (1990) 763.
  • 3,4-Disubstituted g-lactam rongs as conformationally constrained mimics of peptide derivatives containing aspartic acid or norleucine
    Garvey, D.S.; May, P.D.; Nadzan, A.M.; J. Org. Chem., 55 (1990) 936.
  • Synthesis of advanced quinocarcin intermediate from L-glutamic acid
    Lessen, T.A.; Demko, D.M.; Weireb, S.M.; Tetrahedron Lett., 31 (1990) 2105.
  • Synthesis of 7-ethyl-4,7-dihydro-4-oxo-2-(4-pyridinyl)hieno[2,3-b]pyridine-5-carboxylic acid
    Bacon, E.R.; Daum, S.J.; J. Heterocyclic Chem., 28 (1991) 1953.
  • Expanded heterohelicenes: molecular coils that form chiral complexes
    Bell, T.W.; Jousselin, H.; J. Am. Chem. Soc.; 113 (1991) 6283.
  • b-Carbolin-Alkaloide, II. Tributyl(1-ethoxyvinyl)stannan als C2-Baustein für die Synthese von b-Carbolin-Alkaloiden
    Bracher, F.; Hildebrand, D.; Liebigs Ann. Chem., (1993) 837.
  • Enantioselective synthesis of 5-substituted- and 3,5-disubstituted-2-formylpyrrolidine derivatives, the key D-ring fragments of (-)-quinocarcin and (-)-decarboxyquinocarcin
    Katoh, T.; Nagata, Y.; Kobayashi, Y.; Arai, K.; Minami, J.; Tereshima, S.; Tetrahedron Lett., 34 (1993) 5743.
  • Synthesis of 3-(N-alkylamino)acetophenones via a benzyne intermediate
    Albright, J.D.; Liebermann, D.F.; J. Heterocyclic Chem., 31 (1994) 537.
  • Total synthesis of drimane sesquiterpenes from S-(+)-carvone (part 5)
    Swarts, H.J.; Verstegen-Haaksma, A.A.; Jansen B.J.M.; de Groot, A.; Tetrahedron, 50 (1994) 10083.
  • Synthesis and stereochemistry of some thiazolidines related to 6-(hydroxyethyl)-penams
    Urban, F.J.; Bordner, J.; DeCosta, D.; Dee, M.F.; Vincent, L.A.; Tetrahedron: Asymmetry, 5 (1994) 215.
  • The serotonin 5-HT4 receptor. 2. Structure-activity studiem of the indole carbazimidamide class of agonists
    Buchheit, K.-H.; Gamse, R.; Giger, R.; Hoyer, D.; Klein, F.; Kloppner, E.; Pfannkuche, H.-J.; Maties, H.; J. Med. Chem., 38 (1995) 2331.
  • Cyclic variations of 3-quinolinecarboxamides and effects on antiherpetic activity
    Wentland, M.P.; Carlson, J.A.; Dorff, P.H.; Aldous, S.C.; Perni, R.B.; Young, D.C.; Woods, M.G.; Kingsley, S.D.; Ryan, K.A.; Rosi, D.; Drozd, M.L.; Dutko, F.J.; J. Med. Chem., 38 (1995) 2541.
  • Novel and potent adenosine 3',5'-cyclic phosphate phosphodiesterase III inhibitors: thiazolo [4,5-b] [1,6]naphthyridin-2-ones
    Singh, B.; Bacon, E.R.; Lesher, G.Y.; Robinson, S.; Pennock, P.O.; Bode, D.C.; Pagani, E.D.; Bentley, R.G.; Connell, M.J.; Hamel, L.T.; Silve, P.J.; J. Med. Chem., 38 (1995) 2546.
  • New synthetic routes to 3-, 5-, and 6-aryl-2-chloropyridines
    Chuch, R.; Trust, R.; Albright, J.D.; Powell, D.W.; J. Org. Chem., 60 (1995) 3750.
  • Synthesis of functionalized aryloxy 1,3-butadienes and their transformation to diaryl ethers via Diels - Alder cycloaddition reactions
    Olsen, R.K.; Feng, X.; Campbell, M.; Shao, R.; Math, S.K.; J. Org. Chem., 60 (1995) 6025.
  • Mannich biscyclization. Total synthesis of (-)-ajamalicine
    Logers, M.; Ogerman, L.E.; Welmaker, G.S.; J. Am. Chem. Soc.; 117 (1995) 9139.
  • A novel approach to the synthesis of 1-substituted-3,6-diaryl-imidazo[1,5-b]pyridazines
    Zhao, X.; Zhang, R.; Synth. Comm., 25 (1995) 3271.
  • Synthesis of kainoid analogues
    Barraclough, P.; Hudhomme, P.; Spray, C.A.; Young, D.W.; Tetrahedron, 51 (1995) 4195.
  • Stereospecific synthesis of (2S,4R)-[5,5,5-2H3]leucine
    August, R.A.; Khan, J.A.; Moody, C.M.; Young, D.W.; J. Chem. Soc., Perkin Trans. 1, (1996) 507.
  • Study on the preparation of heteroaryl substituted enamines. A simple synthesis of heteroaryl substituted acetaldoximes from enamines
    Copar, A.; Stanovnik, B.; Eisler, M.; J. Heterocyclic Chem., 33 (1996) 465.
  • Concise syntheses of novel 1H-pyrrolo[3,2-g]quinazoline ring system and its [2,3-f] angular isomer
    Showalter, H.D.H.; Sun, L.; Sercel, A.; Winters, R.T.; Denny, W.A.; Palmer, B.D.; J. Org. Chem., 61 (1996) 1155.
  • A novel synthesis of the antipsychotic agent ziprasidone
    Urban, F.J.; Breitenbach, R.; Gonyaw, D.; Synth. Comm., 26 (1996) 1629.
  • Chemistry and nonlinear optical properties of new 2H-benzotriazole derivatives
    Gompper, R.; Walther, P.; Brauchle, C.; Stadle, S.; Tetrahedron, 52 (1996) 14607.
  • Ring contraction of a two-carbon bridged spiropentane
    Wiberg, K.B.; Snoonian, J.R.; Lahti, P.M.; Tetrahedron Lett., 37 (1996) 8285.
  • Synthesis of (h5 -cyclopentadienyl)-1-(4-benzyloxycarbonyl-3,4-dihydroquinoxalin-2-yl )et hene-1,2-dithiolatocobalt(III) and (h5-cyclopentadienyl)-1-[2-(N,N-dimethylaminomethyleneamino)-3-methyl-4-oxopteridin-6-yl]ethene-1,2 -di thiolatocobalt(III)
    Dinsmore, A.; Birks, J.H.; Garner, C.D.; Joule, J.A.; J. Chem. Soc., Perkin Trans. 1, (1997) 801.
  • Synthesis of agonists and antagonists for central glutamate receptors by a novel "ring switching" strategy
    Bowler, A.N.; Dinsmore, A.; Doyle, P.M.; Young, D.W.; J. Chem. Soc., Perkin Trans. 1, (1997) 1297.
  • Nitrosation of methyl 2-cinnamoylamino-3-dimethylaminopropenoates. Alkil N-cinnamoyloxalic acid hydroxyimidic amides, intermediates in the synthesis of alkil 5-styryl-1,2,4-oxodiazole-3-carboxylates
    Kmetic, M.; Stankovik, B.; J. Heterocyclic Chem., 34 (1997) 1705.
  • Synthesis of oligo(diazaphenyls). Tailor-made fluorescent heteroaromatics and pathways to nanostructures
    Gompper, R.; Mair, H.-J.; Polborn, K.; Synthesis, (1997) 696.
  • A convenient and efficient synthesis of (2S,4R)- and (2S,4S)-4-methylglutamic acid
    Coudert, E.; Acher, F.; Azerad, R.; Synthesis, (1997) 863.
  • 4-Substituted protoanemonin in intramolecular cycloaddition reactions of non-stabilised azomethine ylides
    Grigg, R.; Samic, V.; Thornton-Pett, M.; Tetrahedron, 53 (1997) 10633.
  • A convergent route for the total synthesis of the eleuthesides
    Chen, X.-T.; Gutteridge, C.E.; Bhattacharya, S.K.; Zhou, B.; Pettus, T.R.R.; Hascall, T.; Danishefsky, S.J.; Angew. Chem. Int. Ed., 37 (1998) 185.
  • Stereoselective 1,3-Dipolar Cycloadditions to (S)-1-Benzoyl-3-(cyanomethylidene)-5-(methoxycarbonyl)pyrrolidin-2-one
    Skof, M.; Svete, J.; Stanovnik, B.; Golic, L.; Golic-Grdadolnik, S.; Selic, L.; Helv. Chim. Acta, 81 (1998) 2332.
  • Synthesis and structures of 1,3,1',3'-tetrabenzyl-2,2'-biimidazolidinylidenes (electron-rich alkenes), their aminal intermediates and their degradation products
    Çetinkaya, B.; Çetinkaya, E.; Chamizo, J.A.; Hitchcock, P.B.; Jasim, H.A.; Küçükbay, H.; Lappert, M.F.; J. Chem. Soc., Perkin Trans. 1, (1998) 2047.
  • Ring expansion and contraction of a two-carbon bridged spiropentane
    Wilberg, K.W.; Snoonian, J.R.; J. Org. Chem., 63 (1998) 1390.
  • Molecular architecture. 2. Synthesis and metal complexation of heptacyclic terpyridyl molecular clefts
    Bell, T.W.; Cragg, P.J.; Firestone, A.; Kwok, A.D.-I.; Liu, J.; Ludwig, R.; Sodoma, A.; J. Org. Chem., 63 (1998) 2232.
  • 4-(2,2-Dimethyldioxalan-4-yl)-5-(pterin-6-yl)-1,3-dithiol-2-ones proligands relating to the cofactor of the oxomolybdoenzymes
    Dinsmore, A.; Garner, C.D.; Joule, J.A.; Tetrahedron, 54 (1998) 9559.
  • The synthesis and transformations of substituted 2-hydroxy-3-dimethylaminopropenoates. The preparation of condensed 3-hydroxypyran-2-ones
    Smodis, J.; Stanovnik, B.; Tetrahedron, 54 (1998) 9799.
  • Solid phase synthesisof 5-aminopyrazoles and serivatives part II
    Wilson, R.D.; Watson, S.P.; Richards, S.A.; Tetrahedron Lett., 39 (1998) 2827.
  • Spiro-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one derivatives are mixed AMPA and NMDA glycine-site antagonists active in vivo
    Jimonet, P.; Boireau, A.; Chevé, M.; Damour, D.; Genevois-Borella, A.; Imperato, A.; Pratt, J.; Randle, J.C.R.; Ribeill, Y.; Stutzmann, J.-M.; Mignani, S.; Bioorg. Med. Chem. Lett., 9 (1999) 2921.
  • Stereoselective amination of 5-substituted g-lactones and g-lactams - a convenient route for the preparation of 5-substituted (3S,5S)-3-acetylaminotetrahydrofuran-2-ones and (3S,5S)-3-acetylaminopyrrolidin-2-ones
    Skof, M.; Svete, J.; Kmetic, M.; Golic-Grdadolnik, S.; Stanovnik, B.; Eur. J. Org. Chem.; (1999) 1581.
  • Synthesis of Highly Soluble Annelated Polypyridines
    Bejan, E.; Fontenas, C.; Ait-Haddou, H.; Daran, J.-C.; Balavoine, G.G.A.; Eur. J. Org. Chem.; (1999) 2485.
  • The synthesis of methyl 2-(benzyloxycarbonyl)amino-3-dimethylaminopropenoate. The synthesis of trisubstituted pyrroles, 3-amino-2H-pyran-2-ones, Fusem 2H-pyran-2-ones and 4H-pyridin-4-ones
    Toplak, R.; Svete, J.; Stankovnik, B.; Grdadolnik, S.G.; J. Heterocyclic Chem., 36 (1999) 225.
  • Attempts to prepare some 3-substituted azolo[1,2-x]azines, intermediates In the synthesis of azaaplysinopsin derivatives
    Jukic, L.; Copar, A.; Malesic, M.; Krabavcic, A.; Svete, J.; Stankovnik, B.; J. Heterocyclic Chem., 36 (1999) 1147.
  • Regioselective Preparation of N7- and N9-Alkyl Derivatives of N6-[(Dimethylamino)methylene]adenine Bearing an Active Methylene Group and Their Further Derivatization Leading to a-Branched Acyclic Nucleoside Analogues
    Hockova, D.; Budesinsky, M.; Marek, R.; Marek, J.; Holy, A.; Eur. J. Org. Chem.; (1999) 2675.
  • The total synthesis of eleutherobin
    Chen, X.-T.; Bhattacharya, S.K.; Zhou, B.; Gutteridge, C.E.; Pettus, T.R.R.; Danishefsky, S.J.; J. Am. Chem. Soc.; 121 (1999) 6563.
  • Transformations of alkyl 2-(2,2-disubstituted-ethenyl)amino-3-dimethylaminoprop-2-enoates: synthesis of alkyl 3,4-disubstituted- and alkyl 1-acyl-3,4-disubstituted pyrrole-2-carboxylates
    Selic, L.; Stanovnik, B.; Synthesis, (1999) 479.
  • An effective route to polysubstituted symmetric terpyridines
    Sasaki, I.; Daran, J.C.; Balavoine, G.G.A.; Synthesis, (1999) 815.
  • Selective synthesis of b-substituted aspartic acids via tetrahydro-1,3-oxazin-6-ones
    Burtin, G.; Corringer, P.-J.; Hitchcock,P.B.; Young, D.W.; Tetrahedron Lett., 40 (1999) 4275.
    2000 - current date
  • The synthesis and vasopressin (AVP) antagonist activity of a novel series of n-aroyl-2,4,5,6-tetrahydropyrazolo[3,4-d]thieno[3,2-b]azepines
    Albright, J.D.; Santos, E.G.D.; Dusza, J.P.; Chan, P.S.; Coupet, J.; Ru, X.; Mazandarani, H.; Bioorg. Med. Chem. Lett., 10 (2000) 695.
  • Synthesis of New Soluble Annelated Polypyridines
    Ait-Haddou, H.; Fontenas, C.; Bejan, E.; Daran, J.-C.; Balavoine, G.G.A.; Eur. J. Org. Chem.; (2000) 987.
  • Synthesis of (2S)-2-(Benzoylamino)-3-(heteroaryl)propyl Benzoates
    Skof, M.; Svete, J.; Stanovnik, B.; Golic-Grdadolnik, S.; Helv. Chim. Acta, 83 (2000) 760.
  • A Simple Stereoselective Synthesis of Aplysinopsin Analogs
    Selic, L.; Jakse, R.; Lampic, K.; Golic, L.; Golic-Grdadolnik, S.; Stanovnik, B.; Helv. Chim. Acta, 83 (2000) 2802.
  • Tetrahydro-1,3-oxazin-6-ones as templates for the stereoselective synthesis of b-substituted L-aspartic acids
    Burtin, G.; Corringer, P.-J.; Young, D.W.; J. Chem. Soc., Perkin Trans. 1, (2000) 3451.
  • Synthesis of 1,4,5,6-tetrahydropyrazolo[3,4-d]pyrido[3,2-b]azepine
    Albright, J.D.; Du, X.; J. Heterocyclic Chem., 37 (2000) 41.
  • Synthesis of transition state analogue inhibitors for purine nucleoside Phosphorylase and N-ribidose hydrolases
    Evans, G.B.; Furneaux, R.H.; Gainsford, G.J.; Schramm, V.L.; Tyler, P.C.; Tetrahedron, 56 (2000) 3053.
  • New synthesis of 2-aminobicyclo[2.1.1]hexane-2,5-dicarboxylic acid-I (ABHxD-I), a potent metabotropic receptor agonist
    Conti, P.; Kozikowski, A.P.; Tetrahedron Lett., 41 (2000) 4053.
  • Synthetic studiem towards (+)-Dihydroampullicin. Michael addition of N-Boc-2-(tert-butyldimethylsiloxy)-3-methyl-pyrrole to a-methylene lactones
    Marcos, I.; Rudero, E.; Bermejo, F.; Tetrahedron Lett., 41 (2000) 8451.
  • NO-Independent stimulators of soluble guanylate cyclase
    Straub, A.; Stasch, J.-P.; Alonso-Alija, C.; Benet-Buchholz, J.; Ducke, B.; Feurer, A.; Furstner, C.; Bioorg. Med. Chem. Lett., 11 (2001) 781.
  • Synthesis of anticonvulsive AMPA antagonists - 4-Oxo-10-substituted-imidazo[1,2-a]indeno[1,2-e]pyrazin-2-carboxylic acid derivatives
    Stutzmann, J.-M.; Bohme, G.A.; Boireau, A.; Damour, D.; Debono, M.W.; Genevois-Borella, A.; Jimonet, P.; Pratt, J.; Randle, J.C.R.; Ribeill, Y.; Vuilhorgne, M.; Mignani, S.; Bioorg. Med. Chem. Lett., 11 (2001) 1205.
  • 1,3-Dipolar cycloadditions to (5Z)-1-acyl-5-(cyanomethylidene)-imidazolidine-2,4-diones: synthesis and transformations of spirohydantoin derivatives
    Groselj, U.; Drobnic, A.; Recnik, S.; Svete, J.; Stanovnik, B.; Golobic, A.; Lah, N.; Leban, I.; Meden, A.; Golic-Grdadolnik, S.; Helv. Chim. Acta, 84 (2001) 3403.
  • Synthesis of the organic ligand of the molybdenum cofactor, in protected form
    Bradshaw, B.; Dinsmore, A.; Ajana, W.; Collison, D.; Garner, C.D.; Joule, J.A.; J. Chem. Soc., Perkin Trans. 1, (2001) 3239.
  • The synthesis and transformations of 2-[2-ethoxycarbonyl-2-(2-pyridinyl)ethenyl]amino-3-dimethylaminopropenoates. The synthesis of substituted b-amino-a,b-didehydro-a-amino acid derivatives
    Jukic, L.; Recnik, S.; Grdadolnik, S.G.; Svete, J.; Stanovnik, B.; J. Heterocyclic Chem., 38 (2001) 859.
  • Synthesis of (S)-3-heteroaryl-2-hydroxy-1-propyl benzoates by "Ring switching" methodology
    Mihelic, D.; Jakse, R.; Svete, J.; Stanovnik, B.; Grdadolnik, S.G.; J. Heterocyclic Chem., 38 (2001) 1307.
  • A New synthetic router to 3,4-bridged 1,6,6 g4-trithiapentalenes
    Hang, W.; Henry, Y.; Synlett, (2001) 1129.
  • Enaminones acylation: competitive formation of quinolin-4-one and isoquinolin-1-one derivatives
    Vales, M.; Lokshin, V.; Pepe, G.; Samat, A.; Guglielmetti, R.; Synthesis, (2001) 2419.
  • Asymmetric synthesis of a-amino acids from a,b-(Z)-didehydroamino acid derivatives with 1,2,3,6-tetrahydropyrazin-2-one structure
    Abellan, T.; Mancheno, B.; Najera, C.; Sansano, J.M.; Tetrahedron, 57 (2001) 6627.
  • A simple synthesis of aplysinopsin analogues by dimethylamine substitution In N,N-(dimethylamino)methyldiene derivatives of five-membered heterocycles
    Jakse, R.; Recnik, S.; Svete, J.; Golobic, A.; Golic, L.; Stanownik, B.; Tetrahedron, 57 (2001) 8395.
  • Extension of the "ring switch" approach to glutamate antagonists to d-lactam urethanes
    Coe, D.; Drysdale, M.; Philps, O.; West, R.; Young, D.W.; J. Chem. Soc., Perkin Trans. 1, (2002) 2459.
  • Synthesis of spirolactones by 1,3-dipolar cycloadditions to methyl (S)-3-[(E)-cyanomethylidene]-2-oxotetrahydrofuran-5-carboxylate
    Pirc, S.; Recnik, S.; Skof, M.; Svete, J.; Golic, L.; Meden, A.; Stanovnik, B.; J. Heterocyclic Chem., 39 (2002) 411.
  • Synthesis of 1,2-dithiolane analogues of leucine for potential use in peptide chemistry
    Morera, E.; Pinnen, F.; Lucente, G.; Org. Lett., 4 (2002) 1139.
  • An Expedient Synthesis of Highly Functionalized Naphthyridones and Quinolines from a Common N-Aryl Pyridinone Template
    Savarin, C.G.; Murry, J.A.; Dormer, P.G.; Org. Lett., 4 (2002) 2071.
  • Practical synthesis of 8-acyl-7-alkyl-1,6-naphthyridin-5(6H)-ones
    Vales, M.; Lokshin, V.; Pepe, G.; Guglielmetti, R.; Samat, A.; Tetrahedron, 58 (2002) 8543.
  • Stereoselective synthesis of (1R,3R,4R)-3-(1,2,4-triazolo[4,3-x]azin-3-yl)-1,7,7-trimethylbicyclo[2.2.1]heptan-2-ones
    Groselj, U.; Recnik, S.; Svete, J.; Meden, A.; Stanownik, B.; Tetrahedron: Asymmetry, 13 (2002) 821.
  • Novel B-ring modified allocolchicinoids of the NCME series: design, synthesis, antimicrotubule activity and cytotoxicity.
    Bergemann, S.; Brecht, R.; Buttner, F.; Guenard, D.; Gust, R.; Seitz, G.; Stubbs, M.T.; Thoret, S.; Bioorg. Med. Chem., 11 (2003) 1269.
  • Total synthesis of ingenol
    Tanino, K.; Onuki, K.; Asano, K.; Miyashita, M.; Nakamura, T.; Takahashi, Y.; Kuwajima, I.; J. Am. Chem. Soc.; 125 (2003) 1498.
  • Traceless solid phase synthesis of 2-substituted pyrimidines using an "off-the-shelf" chlorogermane-functionalised resin.
    Spivey, A.C.; Srikaran, R.; Diaper, C.M.; Turner, D.J.; Org. Biomom. Chem., 1 (2003) 1638.
  • An alternative to the use of d-lactam urethanes in the "ring switch" approach to higher homologues of AMPA-type glutamate antagonists.
    Hitchcock, P.B.; Masood, S.R.; Young, D.W.; Org. Biomom. Chem., 1 (2003) 2682.
  • Enamine-functionalized oligopyridines as convenient intermediates for the synthesis of carbaldehyde derivatives
    Viau, L.; Senechal, K.; Maury, O.; Guegan, J.-P.; Dupau, P.; Toupet, L.; Le Bozec, H.; Synthesis, (2003) 577.
  • Electrochemical probing of ground state electronic interactions in polynuclear complexes of a new heteroditopic ligand
    Konstable, E.C.; Figgemeier, E.; Housecroft, C.E.; Olsson, J.; Zimmermann, Y.C.; Dalton Trans., (2004) 1918.